Arachidonylcyclopropylamide
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Arachidonylcyclopropylamide
| Arachidonylcyclopropylamide | |
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N-(Cyclopropyl)-5Z,8Z,11Z,14Z-eicosatetraenamide |
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Other names
ACPA |
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| Identifiers | |
| CAS number | 229021-64-1  |
| PubChem | 5311007 |
| ChemSpider | 4470548  |
| ChEMBL | CHEMBL418353 |
| Jmol-3D images | Image 1 |
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| Properties | |
| Molecular formula | C23H37NO |
| Molar mass | 343.55 g mol−1 |
| Solubility in other solvents | soluble in ethanol, chloroform, THF and DMSO |
 Except where noted otherwise, data are given for materials in their standard state (at 25 °C, 100 kPa) |
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| Infobox references | |
Arachidonylcyclopropylamide (ACPA) is a synthetic agonist of the cannabinoid receptor 1 (CB1R). ACPA is considered to be a selective cannabinoid agonist as it binds primarily to the CB1R and has low affinity to the cannabinoid receptor 2 (CB2R) (Ki = 2.2 nM for CB1R; Ki = 700 nM for CB2R). [1]
References
- ^ Hillard, CJ; Manna, S; Greenberg, MJ; Dicamelli, R; Ross, RA; Stevenson, LA; Murphy, V; Pertwee, RG et al (1999). "Synthesis and characterization of potent and selective agonists of the neuronal cannabinoid receptor (CB1)". The Journal of Pharmacology and Experimental Therapeutics 289 (3): 1427–33. PMID 10336536.
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