Agonists: Glutamate/Acite Site Competitive Agonists:
Aspartate •
Glutamate • Homoquinolinic Acid •
Ibotenic Acid •
NMDA •
Quinolinic Acid •
Tetrazolylglycine;
Glycine Site Agonists: ACBD • ACPC • ACPD •
Alanine • CCG •
Cycloserine • DHPG • Fluoroalanine •
Glycine • HA-966 • L-687,414 • Milacemide •
Sarcosine •
Serine •
Tetrazolylglycine;
Polyamine Site Agonists: Acamprosate •
Spermidine •
Spermine
Antagonists: Competitive Antagonists: AP5 (APV) •
AP7 •
CGP-37849 • CGP-39551 • CGP-39653 • CGP-40116 • CGS-19755 • CPP • LY-233,053 • LY-235,959 • LY-274,614 • MDL-100,453 •
Midafotel (d-CPPene) • NPC-12,626 • NPC-17,742 • PBPD •
PEAQX •
Perzinfotel • PPDA • SDZ-220581 •
Selfotel (CGS-19,755);
Noncompetitive Antagonists: ARR-15,896 • FPL-12495 • FR-115,427 •
Hodgkinsine • HU-211 •
Magnesium • MDL-27,266 • NPS-1506 • Psychotridine •
Zinc;
Uncompetitive Pore Blockers: 2-MDP •
8A-PDHQ •
Amantadine •
Aptiganel (CNS-1102) • ARL-12,495 • ARL-15,896-AR • ARL-16,247 •
Budipine •
Delucemine •
Dexoxadrol •
Dieticyclidine •
Dizocilpine (MK-801) • Endopsychosin •
Esketamine •
Etoxadrol •
Eticyclidine •
Gacyclidine •
Ibogaine • Indantadol (CHF-3381) •
Ketamine •
Ketobemidone •
Loperamide •
Memantine •
Meperidine (Pethidine) •
Methadone •
Methorphan (
Dextromethorphan,
Levomethorphan) •
Milnacipran •
Morphanol (
Dextrorphan,
Levorphanol) •
NEFA •
Neramexane •
Nitrous Oxide •
Noribogaine •
Orphenadrine • Phencyclamine •
Phencyclidine •
Propoxyphene •
Remacemide •
Rhynchophylline •
Riluzole •
Rimantadine •
Rolicyclidine •
Tenocyclidine •
Tiletamine •
Tramadol •
Xenon;
Glycine Site Antagonists: ACEA-1021 • ACEA-1328 • ACPC •
Carisoprodol • CGP-39653 • CKA •
DCKA •
Felbamate • Gavestinel (GV-150,526) • GV-196,771 •
Kynurenic Acid • L-689,560 • L-701,324 •
Lacosamide • Licostinel (ACEA-1021) • LU-73,068 • MDL-105,519 •
Meprobamate • MRZ 2/576 • PNQX • ZD-9379;
NR2B Subunit Antagonists: Besonprodil • CO-101,244 (PD-174,494) • CP-101,606 •
Eliprodil •
Haloperidol •
Ifenprodil •
Isoxsuprine •
Nylidrin • Ro8-4304 • Ro25-6981 • Traxoprodil;
Polyamine Site Antagonists: Arcaine • Co 101676 •
Diaminopropane •
Diethylenetriamine •
Huperzine A •
Pentamidine •
Putrescine • Ro 25-6981;
Unclassified/Unsorted Antagonists: Chloroform •
Diethyl Ether •
Enflurane •
Ethanol (Alcohol) •
Halothane •
Isoflurane •
Methoxyflurane
