Brand names: Stadol®, Stadol® NS®
Chemical formula:

- Drug Forms:
- Butorphanol Tartrate Solution for injection (below)
- Butorphanol Tartrate Nasal spray, solution
- Espa�ol:
- Tartrato de butorfanol, Solución para inyección
- Tartrato de Butorfanol Aerosol nasal, solución
Butorphanol Tartrate Solution for injection
What is this medicine?
BUTORPHANOL (byoo TOR fa nole) is a pain reliever. It is used to treat moderate to severe pain. It is also used to prevent pain before surgery and during child birth.
This medicine may be used for other purposes; ask your health care provider or pharmacist if you have questions.
What should I tell my health care provider before I take this medicine?
They need to know if you have any of these conditions:
brain tumor
drug abuse or addiction
head injury
heart disease
if you frequently drink alcohol containing drinks
kidney disease
liver disease
lung or breathing disease, like asthma
an allergic reaction to butorphanol, benzethonium chloride, other medicines, foods, dyes, or preservatives
pregnant or trying to get pregnant
breast-feeding
How should I use this medicine?
This medicine is for injection into a muscle or a vein. It is usually given by a health care professional in a hospital or clinic setting.
If you get this medicine at home, you will be taught how to prepare and give this medicine. Use exactly as directed. Take your medicine at regular intervals. Do not take your medicine more often than directed.
It is important that you put your used needles and syringes in a special sharps container. Do not put them in a trash can. If you do not have a sharps container, call your pharmacist or healthcare provider to get one.
Talk to your pediatrician regarding the use of this medicine in children. This medicine is not approved for use in children.
Overdosage: If you think you have taken too much of this medicine contact a poison control center or emergency room at once.
NOTE: This medicine is only for you. Do not share this medicine with others.
What may interact with this medicine?
Do not take this medicine with any of the following medications:
buprenorphine
nalbuphine
pentazocine
This medicine may also interact with the following medications:
alcohol
antihistamines for allergy, cough and cold
barbiturates, like phenobarbital
medicines for depression, anxiety, or psychotic disturbances
medicines for pain like tramadol and propoxyphene
medicines for sleep
This list may not describe all possible interactions. Give your health care provider a list of all the medicines, herbs, non-prescription drugs, or dietary supplements you use. Also tell them if you smoke, drink alcohol, or use illegal drugs. Some items may interact with your medicine.
What should I watch for while using this medicine?
Tell your doctor or health care professional if your pain does not go away, if it gets worse, or if you have new or a different type of pain. You may develop tolerance to the medicine. Tolerance means that you will need a higher dose of the medicine for pain relief. Tolerance is normal and is expected if you take the medicine for a long time.
Do not suddenly stop taking your medicine because you may develop a severe reaction. Your body becomes used to the medicine. This does NOT mean you are addicted. Addiction is a behavior related to getting and using a drug for a non-medical reason. If you have pain, you have a medical reason to take pain medicine. Your doctor will tell you how much medicine to take. If your doctor wants you to stop the medicine, the dose will be slowly lowered over time to avoid any side effects.
You may get drowsy or dizzy. Do not drive, use machinery, or do anything that needs mental alertness until you know how this medicine affects you. Do not stand or sit up quickly, especially if you are an older patient. This reduces the risk of dizzy or fainting spells. Alcohol may interfere with the effect of this medicine. Avoid alcoholic drinks.
What side effects may I notice from receiving this medicine?
Side effects that you should report to your doctor or health care professional as soon as possible:
allergic reactions like skin rash, itching or hives, swelling of the face, lips, or tongue
anxiety, nervousness, agitation
breathing problems
changes in vision
confusion
feeling faint or lightheaded, falls
irregular or pounding heartbeat
ringing in the ears
Side effects that usually do not require medical attention (report to your doctor or health care professional if they continue or are bothersome):
difficulty sleeping at night
dizziness
drowsiness
dry mouth
loss of appetite
nausea, vomiting
pain at site where injected
This list may not describe all possible side effects. Call your doctor for medical advice about side effects. You may report side effects to FDA at 1-800-FDA-1088.
Where should I keep my medicine?
Keep out of the reach of children. This medicine can be abused. Keep your medicine in a safe place to protect it from theft. Do not share this medicine with anyone. Selling or giving away this medicine is dangerous and against the law.
If you are using this medicine at home, you will be instructed on how to store this medicine. Throw away any unused medicine after the expiration date on the label.
Last updated: 7/1/2002
Important Disclaimer: The drug information provided here is for educational purposes only. It is intended to supplement, not substitute for, the diagnosis, treatment and advice of a medical professional. This drug information does not cover all possible uses, precautions, side effects and interactions. It should not be construed to indicate that this or any drug is safe for you. Consult your medical professional for guidance before using any prescription or over the counter drugs.
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